Frog v1.01.
FRee On line druG conformation
generation.
What is Frog ?
Frog is intended to generate 3D for drugs, usually described using a 1D
or 2D representation. Frog performs isomer identification from
ambiguous compound description. Frog is able to generate
multi-conformations per isomer.
Frog is a tool that results from a collaborative work involving
several teams at RPBS.
Frog
is based on Frowns (http://frowns.sourceforge.net/), a chemoinformatics
toolkit written in python, to which several features have been added.
Frog has some limitations (as almost every other package of the field).
Test used the series of compounds of the
astex diverse test set to evaluate Frog.
The list of the ligands' smiles from this test set, which have been employed as input for the generation of them conformations,
can be accessed
here.
For each ligand, 4 runs of generations were made. Theirs results are listed below.
abreviations:
- meanNc: number of conformations generated over the 4 runs
- minClRmsd: closest RMSD over the 4 runs
- meanClRmsd: mean of the closest RMSD over the 4 runs
- sdClRmsd: standard-deviation of the closest RMSD over the 4 runs
- maxLaRmsd: largest RMSD over the 4 runs
- meanLaRmsd: mean of the largest RMSD over the 4 runs
- sdLaRmsd: standard-deviation of the largest RMSD over the 4 runs
results:
| ligand | nb. atoms | meanNc | minClRmsd | meanClRmsd | sdClRmsd | maxLaRmsd | meanLaRmsd | sdLaRmsd |
| 1g9v | 25 | 50 | 1.20 | 1.31 | 0.12 | 3.03 | 2.96 | 0.09 |
| 1gkc | 22 | 50 | 1.34 | 1.43 | 0.10 | 3.15 | 3.07 | 0.05 |
| 1gm8 | 24 | 50 | 1.05 | 1.09 | 0.04 | 2.83 | 2.76 | 0.05 |
| 1gpk | 18 | 1 | 1.99 | 1.99 | 0.00 | 1.99 | 1.99 | 0.00 |
| 1hnn | 14 | 2 | 0.42 | 0.51 | 0.08 | 1.20 | 1.18 | 0.04 |
| 1hp0 | 19 | 6 | 0.95 | 0.96 | 0.00 | 2.21 | 2.20 | 0.01 |
| 1hq2 | 14 | 3 | 0.15 | 0.26 | 0.15 | 0.57 | 0.57 | 0.00 |
| 1hvy | 32 | 50 | 1.79 | 1.90 | 0.12 | 3.88 | 3.82 | 0.06 |
| 1hwi | 30 | 50 | 0.91 | 1.03 | 0.13 | 3.09 | 3.02 | 0.06 |
| 1hww | 12 | 1 | 0.89 | 0.89 | 0.00 | 0.89 | 0.89 | 0.00 |
| 1ia1 | 19 | 4 | 0.67 | 1.07 | 0.27 | 2.02 | 1.89 | 0.14 |
| 1ig3 | 18 | 26 | 0.76 | 0.78 | 0.02 | 2.37 | 2.29 | 0.06 |
| 1j3j | 17 | 4 | 0.41 | 0.48 | 0.08 | 1.27 | 1.23 | 0.04 |
| 1jd0 | 13 | 12 | 0.57 | 0.57 | 0.00 | 1.48 | 1.37 | 0.12 |
| 1jje | 25 | 50 | 0.95 | 1.11 | 0.11 | 2.63 | 2.57 | 0.05 |
| 1jla | 27 | 50 | 1.00 | 1.15 | 0.11 | 3.07 | 3.04 | 0.04 |
| 1k3u | 21 | 50 | 1.04 | 1.12 | 0.09 | 2.60 | 2.55 | 0.04 |
| 1ke5 | 23 | 36 | 0.61 | 0.67 | 0.05 | 2.34 | 2.30 | 0.06 |
| 1kzk | 41 | 46 | 1.75 | 2.09 | 0.23 | 4.77 | 4.70 | 0.09 |
| 1l2s | 19 | 50 | 0.26 | 0.33 | 0.06 | 2.72 | 2.65 | 0.05 |
| 1l7f | 23 | 27 | 1.19 | 1.25 | 0.05 | 2.66 | 2.36 | 0.33 |
| 1lpz | 32 | 50 | 1.36 | 1.68 | 0.39 | 3.22 | 3.04 | 0.16 |
| 1lrh | 14 | 9 | 0.32 | 0.68 | 0.24 | 1.22 | 1.14 | 0.08 |
| 1m2z | 28 | 9 | 1.70 | 1.72 | 0.01 | 1.91 | 1.87 | 0.03 |
| 1meh | 23 | 8 | 0.80 | 1.19 | 0.26 | 2.55 | 2.48 | 0.06 |
| 1mmv | 15 | 50 | 0.51 | 0.58 | 0.09 | 2.11 | 2.02 | 0.06 |
| 1mzc | 35 | 50 | 1.90 | 2.16 | 0.23 | 3.56 | 3.53 | 0.03 |
| 1n1m | 12 | 18 | 0.73 | 0.83 | 0.07 | 1.89 | 1.85 | 0.03 |
| 1n2j | 10 | 12 | 1.32 | 1.33 | 0.01 | 1.86 | 1.85 | 0.01 |
| 1n2v | 15 | 27 | 0.32 | 0.33 | 0.01 | 1.34 | 1.33 | 0.02 |
| 1n46 | 27 | 4 | 0.99 | 1.47 | 0.37 | 2.38 | 2.26 | 0.11 |
| 1nav | 23 | 32 | 0.73 | 0.86 | 0.24 | 2.67 | 2.62 | 0.04 |
| 1of1 | 18 | 2 | 1.14 | 1.21 | 0.09 | 1.77 | 1.53 | 0.23 |
| 1of6 | 13 | 18 | 0.61 | 0.69 | 0.08 | 1.69 | 1.66 | 0.05 |
| 1opk | 29 | 34 | 0.69 | 0.75 | 0.07 | 2.50 | 2.45 | 0.08 |
| 1oq5 | 26 | 36 | 0.77 | 0.95 | 0.14 | 1.75 | 1.68 | 0.07 |
| 1owe | 22 | 16 | 0.71 | 0.84 | 0.11 | 2.18 | 2.10 | 0.07 |
| 1oyt | 30 | 50 | 1.53 | 1.59 | 0.04 | 3.04 | 2.96 | 0.06 |
| 1p2y | 12 | 3 | 0.93 | 1.35 | 0.28 | 1.57 | 1.54 | 0.06 |
| 1p62 | 18 | 6 | 1.22 | 1.25 | 0.04 | 1.96 | 1.94 | 0.01 |
| 1pmn | 33 | 50 | 0.69 | 0.79 | 0.07 | 2.80 | 2.72 | 0.05 |
| 1q1g | 20 | 26 | 1.05 | 1.08 | 0.03 | 2.42 | 2.42 | 0.00 |
| 1q41 | 21 | 1 | 0.44 | 0.44 | 0.00 | 0.44 | 0.44 | 0.00 |
| 1q4g | 17 | 18 | 0.21 | 0.43 | 0.22 | 1.62 | 1.52 | 0.07 |
| 1r1h | 29 | 50 | 1.61 | 1.78 | 0.20 | 3.07 | 3.01 | 0.06 |
| 1r55 | 23 | 50 | 1.35 | 1.42 | 0.05 | 2.99 | 2.91 | 0.06 |
| 1r58 | 23 | 50 | 1.34 | 1.55 | 0.18 | 3.76 | 3.60 | 0.12 |
| 1r9o | 18 | 12 | 0.21 | 0.47 | 0.17 | 1.77 | 1.71 | 0.05 |
| 1s19 | 30 | 50 | 1.50 | 1.53 | 0.02 | 2.77 | 2.70 | 0.07 |
| 1s3v | 27 | 35 | 0.68 | 1.04 | 0.52 | 3.49 | 3.19 | 0.23 |
| 1sg0 | 17 | 4 | 0.38 | 0.39 | 0.01 | 1.25 | 1.25 | 0.01 |
| 1sj0 | 33 | 50 | 2.08 | 2.24 | 0.11 | 3.79 | 3.51 | 0.45 |
| 1sq5 | 15 | 50 | 1.49 | 1.51 | 0.02 | 2.16 | 2.13 | 0.02 |
| 1sqn | 22 | 1 | 1.56 | 1.56 | 0.00 | 1.56 | 1.56 | 0.00 |
| 1t40 | 28 | 50 | 1.20 | 1.32 | 0.12 | 3.26 | 3.20 | 0.06 |
| 1t46 | 37 | 50 | 1.24 | 1.52 | 0.24 | 4.05 | 3.98 | 0.10 |
| 1t9b | 23 | 33 | 0.56 | 0.79 | 0.22 | 2.59 | 2.56 | 0.03 |
| 1tow | 19 | 50 | 0.58 | 0.65 | 0.06 | 1.81 | 1.72 | 0.08 |
| 1tt1 | 15 | 50 | 1.53 | 1.53 | 0.00 | 2.02 | 2.01 | 0.01 |
| 1tz8 | 20 | 36 | 0.30 | 0.45 | 0.11 | 1.62 | 1.59 | 0.02 |
| 1u1c | 20 | 50 | 0.44 | 0.50 | 0.04 | 2.37 | 2.32 | 0.05 |
| 1u4d | 18 | 1 | 0.14 | 0.23 | 0.18 | 0.51 | 0.23 | 0.18 |
| 1uml | 33 | 50 | 1.04 | 1.37 | 0.35 | 4.07 | 3.96 | 0.08 |
| 1unl | 26 | 50 | 0.91 | 1.05 | 0.14 | 2.59 | 2.42 | 0.19 |
| 1uou | 16 | 9 | 0.91 | 1.00 | 0.07 | 1.88 | 1.85 | 0.06 |
| 1v0p | 30 | 50 | 0.78 | 0.92 | 0.11 | 3.48 | 3.41 | 0.07 |
| 1v48 | 22 | 50 | 0.80 | 0.89 | 0.11 | 2.62 | 2.47 | 0.11 |
| 1v4s | 23 | 18 | 0.50 | 0.94 | 0.46 | 2.84 | 2.79 | 0.07 |
| 1vcj | 25 | 50 | 0.49 | 0.62 | 0.09 | 1.82 | 1.80 | 0.03 |
| 1w1p | 11 | 1 | 0.41 | 0.41 | 0.00 | 0.41 | 0.41 | 0.00 |
| 1w2g | 17 | 6 | 0.99 | 1.00 | 0.01 | 1.67 | 1.63 | 0.03 |
| 1x8x | 13 | 18 | 0.55 | 0.58 | 0.03 | 1.72 | 1.70 | 0.02 |
| 1xm6 | 19 | 33 | 0.42 | 0.62 | 0.20 | 2.14 | 2.10 | 0.04 |
| 1xoq | 26 | 50 | 0.69 | 0.82 | 0.12 | 2.87 | 2.65 | 0.16 |
| 1xoz | 29 | 3 | 1.25 | 1.47 | 0.44 | 2.47 | 1.90 | 0.38 |
| 1y6b | 34 | 50 | 0.61 | 0.73 | 0.13 | 4.05 | 3.69 | 0.27 |
| 1ygc | 38 | 50 | 1.32 | 1.56 | 0.20 | 4.78 | 4.38 | 0.40 |
| 1yqy | 23 | 50 | 1.08 | 1.12 | 0.03 | 3.21 | 3.04 | 0.12 |
| 1yv3 | 22 | 2 | 0.52 | 0.52 | 0.00 | 0.88 | 0.70 | 0.21 |
| 1yvf | 28 | 47 | 1.10 | 1.17 | 0.07 | 3.10 | 3.08 | 0.02 |
| 1ywr | 35 | 50 | 0.96 | 1.13 | 0.22 | 3.54 | 3.43 | 0.10 |
| 1z95 | 29 | 50 | 1.05 | 1.21 | 0.16 | 3.00 | 2.98 | 0.03 |
| 2bm2 | 30 | 50 | 1.34 | 1.51 | 0.14 | 3.69 | 3.57 | 0.09 |
| 2br1 | 29 | 50 | 0.67 | 0.71 | 0.06 | 1.72 | 1.71 | 0.01 |
| 2bsm | 27 | 50 | 0.51 | 0.62 | 0.11 | 2.27 | 2.13 | 0.13 |
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